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- Acetylon Pharmaceuticals, Inc.
- Algomedix, Inc.
- ASINEX
- AsisChem, Inc.
- BioSeek, Inc.
- Broad Institute
- Cedars-Sinai Medical Center
- ChemBridge Corporation
- Columbia University
- Consejo Superior de Investigaciones Cientificas (CSIC), Instituto de Parasitologia y Biomedicina "Lopez-Neyra", Spain
- Cornell University
- Drugs for Neglected Diseases initiative
- Fred Hutchinson Cancer Research Center
- GlaxoSmithKline
- Harvard University
- Indiana University
- Indiana University-Purdue University Indianapolis
- Institut Pasteur de Montevideo, Uruguay
- Johns Hopkins University
- Longevica Pharmaceuticals, Inc.
- Louisiana State University-Health Sciences Center
- LITMUS, LLC
- Marine Biological Laboratory
- Massachusetts Institute of Technology
- Melior Discovery, Inc.
- MOLISA GmbH, Germany
- Myelin Repair Foundation
- NIMH Psychoactive Drug Screening Program
- Numerate, Inc.
- Northeastern University
- Northwestern University
- Ohio State University
- PharmSelex
- Public Library of Science
- Purdue University
- The Rockefeller University
- San Francisco VA Medical Center
- Scripps Research Institute
- Seattle Biomedical Research Institute
- Semafore Pharmaceuticals, Inc.
- St. Jude Children's Research Hospital
- Stanford University
- STATegics, Inc.
- TimTec, Inc.
- Torrey Pines Institute for Molecular Studies
- UCSF General Hospital
- University of California, Berkeley
- University of California, Davis
- University of California, Los Angeles
- University of California, San Diego
- University of California, San Francisco
- University of California, Santa Cruz
- University of Cape Town, South Africa
- University of Cincinnati
- University of Dundee, Scotland
- University of Georgia
- University of Mississippi
- University of North Carolina
- University of Pennsylvania
- University of Pittsburgh
- University of Sydney, Australia
- University of Texas
- University of Washington